Dermorphin 10mg Bottle Already Pain Killer Morphine Replacement Peptide Hormone Strong Analgesic
dermorfina
No CAS: 77614-16-5
Fórmula molecular: C40H50N8O10
Peso molecular: 802.89
Forma: Hormona peptídica Dermorphin lista en 10 mg/vial. un analgésico fuerte.
Dermorphin 10mg/vial
La dermorfina es un heptapéptido aislado por primera vez de la piel de ranas sudamericanas pertenecientes al género Phyllomedusa.. El péptido es un opioide natural que se une como agonista con alta potencia y selectividad a los receptores opioides mu.
Dermorphin is about 30-40 times more potent than morphine but theoretically may be less likely to produce drug tolerance and addiction (due to its high potency). The amino acid sequence of dermorphin is H-Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NH2.
Dermorphin is not found in humans or other mammals and similar D-amino acid peptides have only been found in bacteria, amphibians and molluscs. Dermorphin appears to be made in these through an unusual posttranslational modification carried out by an amino acid isomerase. This unusual process is needed because the D-alanine in this peptide is not among the 20 amino acids coded for in the genetic code and thus the peptide cannot be synthesized in the usual way from the encodings in the genome of an organism.
Dermorphin has been illegally used in horse racing as a performance-enhancing drug. Due to dermorphin’s painkilling activity, horses treated with dermorphin may run harder than they would otherwise.
