Dermorphin 10mg Bottle Already Pain Killer Morphine Replacement Peptide Hormone Strong Analgesic
Dermorfina
Nr CAS: 77614-16-5
Formuła molekularna: C40H50N8O10
Waga molekularna: 802.89
Formularz: Hormon peptydowy Dermorphin gotowy w 10mg/fiolkę. silny środek przeciwbólowy.
Dermorphin 10mg/vial
Dermorphin to hepta-peptyd wyizolowany po raz pierwszy ze skóry południowoamerykańskich żab należących do rodzaju Phyllomedusa. Peptyd jest naturalnym opioidem, który wiąże się jako agonista o dużej sile i selektywności z receptorami opioidowymi mu.
Dermorphin is about 30-40 times more potent than morphine but theoretically may be less likely to produce drug tolerance and addiction (due to its high potency). The amino acid sequence of dermorphin is H-Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NH2.
Dermorphin is not found in humans or other mammals and similar D-amino acid peptides have only been found in bacteria, amphibians and molluscs. Dermorphin appears to be made in these through an unusual posttranslational modification carried out by an amino acid isomerase. This unusual process is needed because the D-alanine in this peptide is not among the 20 amino acids coded for in the genetic code and thus the peptide cannot be synthesized in the usual way from the encodings in the genome of an organism.
Dermorphin has been illegally used in horse racing as a performance-enhancing drug. Due to dermorphin’s painkilling activity, horses treated with dermorphin may run harder than they would otherwise.
